3. Note: The above intermediates are not for sales where the Patents are applicable & still valid.
Intermediates under Development
S. No. Product Name Stage CAS No. Chemical Name
1 Aliskiren ALN01 173336-76-0 4-Bromo-1-methoxy-2(3-methoxypropoxy) benzene
ALN07 Not Available (2S,7S)-2-isopropyl-7-{4-methoxy-3-(3-
methoxypropoxy)bezyl}-8-methylnonayl-N,N-
dimethylformamide
ALN08 Not Available (S)-2-[(S)-2-bromo-2-((2R,4S)-4-isopropyl-5-oxo-
tetrahydrofuran-2-yl)-ethyl-1-[3-(3-methoxy propoxy)-4-
methylphenyl] -3-methylbutyl ester
ALN10 Not Available (2S,4S,5S,7S)-5-azido-4-hydroxy-2-isopropy-7-[4-
methoxypropoxy)-benzyl]-8-methyl nonanic acid (2-
carbamoyl-2-methyl propyl) amide
AL10 Not Available 2(S)-(tert-butoxycarbonyl)amino-4(S)-isopropyl-5-(p-tert-
butyl-phenyl)-pentanal.
2 Ezetimibe EB02 Not Available (4S)-3-[(5S)-5-(4-fluorophenyl)-5-hydroxy pentanoyl]-4-
phenyl-1,3- oxazolidin-2-one
EB03 Not Available (S)-3-{(R)-2-[(S)-4-(trimethylsilyloxy)-phenyl]-(4-
fluorophenylamine)-methyl -4-[2-(4-fluorophenyl)-(1S)-
trimethyl silyloxy]-butyric}-4-phenyl-oxazolidine-2-one
4. EB04 Not Available (3R,4S)-1-(4-Fluorophenyl)-3-[(3S)-3-
(4-fluorophenyl)-3-(trimethylsilyloxy) propyl]-4-(4-
(trimethylsilyloxy)phenyl)-2-azetidinone
EZ04 Not Available (3R,4S)-1-(4-Fluorophenyl)-3-[3-(hydroxy)-3-
oxopropyl]-4-(4-benzyloxyphenyl)-2-azetidonone
3 Eletriptan EL06 Not Available 5-[2-(Benzene sulfonyl)ethenyl]-3-(1-methyl
pyrrolidin-2(R)yl methyl)-1H-indole
4 Linezolid LZN04 Not Available (5R)-5-(chloromethyl)-3-[3-fluoro-4-(4-
morpholinyl)phenyl]-2-oxazolidinone
LZN05 Not Available (S)-N-[[3-[3-Fluoro-4-[4-morpholinyl]phenyl]-2-oxo-5-
oxazolidinyl]methyl]pthalamide
5 Quetiapine QTS01 13349-82-1 1-[2-(2-Hydroxyethoxy) ethyl]piperazine
6 Valsartan -- 195435-23-5 (R)-3-Methyl-2-(N-((2`-(2-trityl -2H-tetrazol-5-
yl)biphenyl-4-yl) methyl)pentananamido) butanoic acid
OR Trityl valsartan
-- 137863-20-8 N-[2`-(1H-tetrazol-5-yl)biphenyl-4-yl methyl]-N-Valeryl-
(L)-valine benzyl ester OR Valsartan benzyl ester
7 Ziprasidone Int -I 118289-55-7 5-(2-chloroethyl)-6-chlorooxindole
Int - II 144010-02-6 3-(1-Piperazinyl)-1,2- benzisothiazole hydrochloride
Note: The above intermediates are not for sales where the Patents are applicable & still valid.